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Þorsteinn Loftsson - Professor Emeritus
–
School of Health Sciences
Þorsteinn Loftsson
Íslenska
Professor Emeritus
Location
Hagi / Ha-313
Phone
525 - 4464
Email
thorstlo [at] hi.is
Unit
Faculty of Pharmaceutical Sciences
Published Work
Þorsteinn Loftsson - published work
Curriculum Vitae
Þorsteinn Loftsson - Curriculum Vitae
ORCID site
https://orcid.org/0000-0002-9439-1553
Research portal – Þorsteinn Loftsson
Under construction throughout the autumn semester 2023
Collaboration
Lipid Pharmaceuticals, Reykjavik, Iceland.
,
Lipid Pharmaceuticals, Reykjavik, Iceland.
Oculis ehf., Reykjavik, Iceland.
,
Oculis ehf., Reykjavik, Iceland.
Prof. Einar Stefánsson
,
Dept. of Medicine, University of Iceland.
Education
0
,
Ph.D.
,
University of Kansas
,
Ph.D.
0
,
MS
,
University of Kansas
,
MS
0
,
MS
,
University of Copenhagen
,
M.S. Pharm. degree
Professional Experience
1986 -
,
Professor of Physical Pharmacy,
University of Iceland in Reykjavik, Iceland
1983 -
1985,
Associate Professor,
University of Iceland
1979 -
1983,
Assistant Professor,
University of Iceland
Published works
2023
Anomalous Properties of Cyclodextrins and Their Complexes in Aqueous Solutions
Materials
Voriconazole Eye Drops: Enhanced Solubility and Stability through Ternary Voriconazole/Sulfobutyl Ether β-Cyclodextrin/Polyvinyl Alcohol Complexes
International Journal of Molecular Sciences
Topical dexamethasone delivery to the retina: An aqueous cyclodextrin-based microsuspension
Journal of Drug Delivery Science and Technology
2022
Stabilization and solubilization of difluprednate in aqueous cyclodextrin solution and its characterization for ophthalmic delivery
Journal of Drug Delivery Science and Technology
Development of Fenofibrate/Randomly Methylated β-Cyclodextrin-Loaded Eudragit® RL 100 Nanoparticles for Ocular Delivery
Molecules
Effect of salt formation on γ-cyclodextrin solubilization of irbesartan and candesartan and the chemical stability of their ternary complexes
Journal of Drug Delivery Science and Technology
Cyclodextrins and Drug Membrane Permeation: Thermodynamic Considerations
Journal of Pharmaceutical Sciences
Aqueous eye drops containing drug/cyclodextrin nanoparticles deliver therapeutic drug concentrations to both anterior and posterior segment
Acta Ophthalmologica
Aqueous Prostaglandin Eye Drop Formulations
Pharmaceutics
A Current Overview of Cyclodextrin-Based Nanocarriers for Enhanced Antifungal Delivery
Pharmaceuticals
Structural Characterization Study of a Lipid Nanocapsule Formulation Intended for Drug Delivery Applications Using Small-Angle Scattering Techniques
Molecular Pharmaceutics
Physicochemical and Stability Evaluation of Topical Niosomal Encapsulating Fosinopril/γ-Cyclodextrin Complex for Ocular Delivery
Pharmaceutics
2021
Bio-Distribution and Pharmacokinetics of Topically Administered γ-Cyclodextrin Based Eye Drops in Rabbits
Pharmaceuticals
Cytotoxicity of β-Cyclodextrins in Retinal Explants for Intravitreal Drug Formulations
Molecules
1,4-Benzodiazepines: Chemical stability and cyclodextrin solubilization
Journal of Drug Delivery Science and Technology
2020
Characterization and Evaluation of Ternary Complexes of Ascorbic Acid with γ-Cyclodextrin and Poly(vinyl Alcohol)
International Journal of Molecular Sciences
Effect of porcine pancreatic α-amylase on dexamethasone release from aqueous solution containing natural γ-cyclodextrin
International Journal of Pharmaceutics
Antifungal activity of econazole nitrate/cyclodextrin complex: Effect of pH and formation of complex aggregates
International Journal of Pharmaceutics
Stability characterization, kinetics and mechanism of tacrolimus degradation in cyclodextrin solutions
International Journal of Pharmaceutics
In Vitro and Ex Vivo Evaluation of Nepafenac-Based Cyclodextrin Microparticles for Treatment of Eye Inflammation
Nanomaterials
2019
Drug delivery to retinal photoreceptors
Drug Discovery Today
Cyclodextrin–Amphiphilic Copolymer Supramolecular Assemblies for the Ocular Delivery of Natamycin
Nanomaterials
Nepafenac-Loaded Cyclodextrin/Polymer Nanoaggregates: A New Approach to Eye Drop Formulation
Materials
Interaction of Native Cyclodextrins and Their Hydroxypropylated Derivatives with Carbamazepine in Aqueous Solution. Evaluation of Inclusion Complexes and Aggregates Formation
ACS Omega
Self-association of cyclodextrins and cyclodextrin complexes in aqueous solutions
International Journal of Pharmaceutics
2018
Self-assembled cyclodextrin-based nanoparticles for meropenem stabilization
Journal of Drug Delivery Science and Technology
2-Hydroxypropyl-β-Cyclodextrin Aggregates: Identification and Development of Analytical Techniques
Materials
Novel excipients – Regulatory challenges and perspectives – The EU insight
International Journal of Pharmaceutics
Topical drug delivery to the posterior segment of the eye: The effect of benzalkonium chloride on topical dexamethasone penetration into the eye in vivo
Journal of Drug Delivery Science and Technology
Solubility of Cyclodextrins and Drug/Cyclodextrin Complexes
Molecules
Topical drug delivery to the posterior segment of the eye: Dexamethasone concentrations in various eye tissues after topical administration for up to 15 days to rabbits
Journal of Drug Delivery Science and Technology
Disruption of α- and γ-cyclodextrin aggregates promoted by chaotropic agent (urea)
Journal of Drug Delivery Science and Technology
2015
Formation and stability assessment of self-assembled nanoparticles from large Mw chitosan and sulfobutylether-β-cyclodextrin
Journal of Drug Delivery Science and Technology
2013
Triclosan-loaded with high encapsulation efficiency into PLA nanoparticles coated with β-cyclodextrin polymer
Journal of Inclusion Phenomena and Macrocyclic Chemistry
Encapsulation of drug molecules into Calix[n]arene Nanobaskets. Role of Aminocalix[n]arenes in biopharmaceutical field
Journal of Pharmaceutical Sciences
Dextran-based cyclodextrin polymers: Their solubilizing effect and self-association
Carbohydrate Polymers
A permeation method for detection of self-aggregation of doxorubicin in aqueous environment
International Journal of Pharmaceutics
For the special IJP issue "Poorly soluble drugs"
International Journal of Pharmaceutics
Physicochemical characterization and stability of microbeads containing cod-liver oil encircled with natural cyclodextrins
Journal of Inclusion Phenomena and Macrocyclic Chemistry
Antifungal drug solubilizing activity and self-aggregation ability of cationic aminocalix[4]arene in comparison to SBEβCD: effect of addition of water-soluble polymer
Journal of Inclusion Phenomena and Macrocyclic Chemistry
Dexamethasone eye drops containing γ-cyclodextrin-based nanogels
International Journal of Pharmaceutics
Cyclodextrins
International Journal of Pharmaceutics
2012
Cyclodextrin-based nanogels for pharmaceutical and biomedical applications
International Journal of Pharmaceutics
Self-assembly of cyclodextrins: Formation of cyclodextrin polymer based nanoparticles
Journal of Drug Delivery Science and Technology
Drug permeation through biomembranes: Cyclodextrins and the unstirred water layer
Pharmazie
Clinical trial: Marine lipid suppositories as laxatives
Marine Drugs
Cyclodextrins as functional excipients: Methods to enhance complexation efficiency
Journal of Pharmaceutical Sciences
Topical drug delivery to the eye: Dorzolamide
Acta Ophthalmologica
The effect of parenterally administered cyclodextrins on the pharmacokinetics of coadministered drugs
Journal of Pharmaceutical Sciences
Cross-linked hydroxypropyl-β-cyclodextrin and γ-cyclodextrin nanogels for drug delivery: Physicochemical and loading/release properties
Carbohydrate Polymers
2011
Self-assembly of cyclodextrin complexes: Effect of temperature, agitation and media composition on aggregation
International Journal of Pharmaceutics
Self-assembly of cyclodextrin complexes: Aggregation of hydrocortisone/cyclodextrin complexes
International Journal of Pharmaceutics
Self-assembly of cyclodextrins: The effect of the guest molecule
International Journal of Pharmaceutics
Drug loading in cyclodextrin polymers: Dexamethasone model drug
Journal of Inclusion Phenomena and Macrocyclic Chemistry
Drug/cyclodextrin: Beyond inclusion complexation
Journal of Inclusion Phenomena and Macrocyclic Chemistry
Pharmaceutical applications of cyclodextrins: Effects on drug permeation through biological membranes
Journal of Pharmacy and Pharmacology
Evaluation of sugammadex self-association
International Journal of Pharmaceutics
Preface: First European cyclodextrin conference
Journal of Inclusion Phenomena and Macrocyclic Chemistry
Topical dexamethasone-cyclodextrin microparticle eye drops for diabetic macular edema
Investigative Ophthalmology and Visual Science
2010
Enalaprilat and enalapril maleate eyedrops lower intraocular pressure in rabbits
Acta Ophthalmologica
Evaluation of a cationic calix[4]arene: Solubilization and self-aggregation ability
International Journal of Pharmaceutics
Effects of cogrinding with β-cyclodextrin on the solid state fentanyl
Journal of Pharmaceutical Sciences
Pharmaceutical applications of cyclodextrins: Basic science and product development
Journal of Pharmacy and Pharmacology
Solubility and permeability of steroids in water in the presence of potassium halides
Pharmazie
γCD/HPγCD mixtures as solubilizer: Solid-state characterization and sample dexamethasone eye drop suspension
Journal of Pharmacy and Pharmaceutical Sciences
Cyclodextrin solubilization of carbonic anhydrase inhibitor drugs: Formulation of dorzolamide eye drop microparticle suspension
European Journal of Pharmaceutics and Biopharmaceutics
Parenteral delivery of HPβCD: Effects on drug-HSA binding
AAPS PharmSciTech
Aqueous solubility and true solutions
Pharmazie
γ-Cyclodextrin hydrogels and semi-interpenetrating networks for sustained delivery of dexamethasone
Carbohydrate Polymers
Effect of self-aggregation of γ-cyclodextrin on drug solubilization
Journal of Inclusion Phenomena and Macrocyclic Chemistry
Self-assembled cyclodextrin aggregates and nanoparticles
International Journal of Pharmaceutics
Cyclodextrins as solubilizers: Formation of complex aggregates
Journal of Pharmaceutical Sciences
Studies of curcumin and curcuminoids. XXXVI. The stoichiometry and complexation constants of cyclodextrin complexes as determined by the phase-solubility method and UV-Vis titration
Journal of Inclusion Phenomena and Macrocyclic Chemistry
2009
Cyclodextrins and their use in pharmacy and cosmetology | Les cyclodextrines et leurs utilisations en pharmacie et cosmétologie
S.T.P. Pharma Pratiques
Fish skin as a model membrane: Structure and characteristics
Journal of Pharmacy and Pharmacology
CDs as solubilizers: Effects of excipients and competing drugs
International Journal of Pharmaceutics
Crystal structure of fentanyl base
X-ray Structure Analysis Online
Drug targeting to the hair follicles: A cyclodextrin-based drug delivery
AAPS PharmSciTech
Diffusion characteristics of vitreous humour and saline solution follow the Stokes Einstein equation
Graefe's Archive for Clinical and Experimental Ophthalmology
2008
Physicochemical properties of water and its effect on drug delivery. A commentary
International Journal of Pharmaceutics
γCD/HPγCD: Synergistic solubilization
International Journal of Pharmaceutics
Comparative interaction of 2-hydroxypropyl-β-cyclodextrin and sulfobutylether-β-cyclodextrin with itraconazole: Phase-solubility behavior and stabilization of supersaturated drug solutions
European Journal of Pharmaceutical Sciences
Topical drug delivery to the posterior segment of the eye: Anatomical and physiological considerations
Pharmazie
Carvedilol: Solubilization and cyclodextrin complexation: A technical note
AAPS PharmSciTech
2007
Development of octanol membranes for drug screening
Journal of Inclusion Phenomena and Macrocyclic Chemistry
Cyclodextrins and their pharmaceutical applications
International Journal of Pharmaceutics
Cyclodextrin microparticles for drug delivery to the posterior segment of the eye: Aqueous dexamethasone eye drops
Journal of Pharmacy and Pharmacology
Cyclodextrins as pharmaceutical solubilizers
Advanced Drug Delivery Reviews
Effects of various cyclodextrins on the stability of freeze-dried lactate dehydrogenase
Journal of Pharmaceutical Sciences
Effects of cyclodextrins on drug delivery through biological membranes
Journal of Pharmaceutical Sciences
Effect of the unstirred water layer on permeability enhancement by hydrophilic cyclodextrins
International Journal of Pharmaceutics
Topical and systemic absorption in delivery of dexamethasone to the anterior and posterior segments of the eye
Acta Ophthalmologica Scandinavica
Studies on curcumin and curcuminoids. XXXI. Symmetric and asymmetric curcuminoids: Stability, activity and complexation with cyclodextrin
International Journal of Pharmaceutics
Antibacterial activity of methylated chitosan and chitooligomer derivatives: Synthesis and structure activity relationships
European Polymer Journal
Cyclodextrins and the liquid-liquid phase distribution of progesterone, estrone and prednicarbate
Journal of Inclusion Phenomena and Macrocyclic Chemistry
Dexamethasone delivery to posterior segment of the eye
Journal of Inclusion Phenomena and Macrocyclic Chemistry
The complexation efficiency
Journal of Inclusion Phenomena and Macrocyclic Chemistry
Cyclodextrins in ocular drug delivery: Theoretical basis with dexamethasone as a sample drug
Journal of Drug Delivery Science and Technology
2006
Determination of aqueous solubility by heating and equilibration: a technical note.
AAPS PharmSciTech [electronic resource].
Influence of aqueous diffusion layer on passive drug diffusion from aqueous cyclodextrin solutions through biological membranes
Pharmazie
Intranasal midazolam: A comparison of two delivery devices in human volunteers
Journal of Pharmacy and Pharmacology
Development and evaluation of an artificial membrane for determination of drug availability
International Journal of Pharmaceutics
The Stokes-Einstein equation and the physiological effects of vitreous surgery
Acta Ophthalmologica Scandinavica
Assessment of mucoadhesion by a resonant mirror biosensor
International Journal of Pharmaceutics
Determination of aqueous solubility by heating and equilibration: A technical note
AAPS PharmSciTech
Ocular powder: Dry topical formulations of timolol are well tolerated in rabbits
Journal of Ocular Pharmacology and Therapeutics
Investigation of soft long chain quaternary ammonium compounds as co-factors to enhance in vitro gene delivery
Pharmazie
Comparison of topical 0.7% dexamethasone-cyclodextrin with 0.1% dexamethasone sodium phosphate for postcataract inflammation
Graefe's Archive for Clinical and Experimental Ophthalmology
2005
Investigation of drug-cyclodextrin complexes by a phase-distribution method: Some theoretical and practical considerations
Chemical and Pharmaceutical Bulletin
Evaluation of cyclodextrin solubilization of drugs
International Journal of Pharmaceutics
Cyclodextrin solubilization of the antibacterial agents triclosan and triclocarban: Formation of aggregates and higher-order complexes
International Journal of Pharmaceutics
Hydrolysis kinetics and QSAR investigation of soft antimicrobial agents
Journal of Pharmacy and Pharmacology
Cyclodextrin solubilization of the antibacterial agents triclosan and triclocarban: Effect of ionization and polymers
Journal of Inclusion Phenomena
Cyclodextrins in drug delivery
Expert Opinion on Drug Delivery
Cyclodextrin formulation of dorzolamide and its distribution in the eye after topical administration
Journal of Controlled Release
2004
Marine lipids as building blocks for soft quaternary ammonium compounds and their antibacterial activity
Pharmazie
Self-Association of Cyclodextrins and Cyclodextrin Complexes
Journal of Pharmaceutical Sciences
Preparation of solid drug/cyclodextrin complexes of acidic and basic drugs
Pharmazie
Synthesis and Characterization of Chitosan N-betainates Having Various Degrees of Substitution
Macromolecules
Applications of chemically-modified cyclodextrins: Use of hydroxypropyl-β-cyclodextrin as an enabling excipient for brain targeting, redox-based derivatives of estradiol: A review of preclinical and clinical findings
Journal of Drug Delivery Science and Technology
The effects of water-soluble polymers on cyclodextrins and cyclodextrin solubilization of drugs
Journal of Drug Delivery Science and Technology
Role of cyclodextrins in improving oral drug delivery
American Journal of Drug Delivery
2003
Examination of 19F-NMR as a tool for investigation of drug-cyelodextrin complexes
Drug Development and Industrial Pharmacy
The effects of cyclodextrins on topical delivery of hydrocortisone: The aqueous diffusion layer
S.T.P. Pharma Sciences
The effects of organic salts on the cyclodextrin solubilization of drugs
International Journal of Pharmaceutics
Investigation and physicochemical characterization of vinpocetine- sulfobutyl ether β-cyclodextrin binary and ternary complexes
Chemical and Pharmaceutical Bulletin
Soft antibacterial agents
Current Medicinal Chemistry
Sublingual delivery of 17β-estradiol from cyclodextrin containing tablets
Pharmazie
Soft antimicrobial agents: Synthesis and activity of labile environmentally friendly long chain quaternary ammonium compounds
Journal of Medicinal Chemistry
2002
Cycloserine fatty acid derivatives as prodrugs: Synthesis, degradation and in Vitro skin permeability
Chemical and Pharmaceutical Bulletin
Mucoadhesive sustained drug delivery system based on cationic polymer and anionic cyclodextrin/triclosan complex
Journal of Inclusion Phenomena
Self association and cyclodextrin solubilization of NSAIDs
Journal of Inclusion Phenomena
Cyclodextrins in eye drop formulations
Journal of Inclusion Phenomena
The effects of cyclodextrins on hydrocortisone permeability through semi-permeable membranes
Journal of Inclusion Phenomena
Self-association and cyclodextrin solubilization of drugs
Journal of Pharmaceutical Sciences
Studies of curcumin and curcuminoids. XXVII. Cyclodextrin complexation: Solubility, chemical and photochemical stability
International Journal of Pharmaceutics
Buccal absorption of ergotamine tartrate using the bioadhesive tablet system in guinea-pigs
International Journal of Pharmaceutics
Cyclodextrins in eye drop formulations: Enhanced topical delivery of corticosteroids to the eye
Acta Ophthalmologica Scandinavica
The use of chemically modified cyclodextrins in the development of formulations for chemical delivery systems
Pharmazie
Cyclodextrins and drug permeability through semi-permeable cellophane membranes
International Journal of Pharmaceutics
Cyclodextrins and the biopharmaceutics classification system of drugs
Journal of Inclusion Phenomena
Fish skin as a model membrane to study transmembrane drug delivery with cyclodextrins
Journal of Inclusion Phenomena
Preface
Journal of Inclusion Phenomena
2001
Sustained drug delivery system based on a cationic polymer and an anionic drug/cyclodextrin complex
Pharmazie
Cyclodextrin solubilization of benzodiazepines: Formulation of midazolam nasal spray
International Journal of Pharmaceutics
Cyclodextrins in topical drug formulations: Theory and practice
International Journal of Pharmaceutics
Intranasal administration of midazolam in a cyclodextrin based formulation: Bioavailability and clinical evaluation in humans
Pharmazie
2000
Methazolamide 1% in cyclodextrin solution lowers IOP in human ocular hypertension
Investigative Ophthalmology and Visual Science
Lipophilic metronidazole derivatives and their absorption through hairless mouse skin
Pharmazie
Marine lipids for prodrugs, soft compounds and other pharmaceutical applications
Pharmazie
Dermal delivery of ETH-615, a zwitterionic drug
Drug Development and Industrial Pharmacy
1999
Cyclodextrins as permeation enhancers: Some theoretical evaluations and in vitro testing
Journal of Controlled Release
Drug-cyclodextrin complexation in the presence of water-soluble polymers: Enhanced solubility and percutaneous transport
ACS Symposium Series
Effect of cyclodextrins and polymers on triclosan availability and substantivity in toothpastes in vivo
Journal of Pharmaceutical Sciences
Diacyl glyceryl ester prodrugs for slow release in the skin: Synthesis and in vitro degradation and absorption studies for naproxen derivatives
Pharmazie
Pharmaceutical applications of β-cyclodextrin
Pharmaceutical Technology
Influence of cyclodextrins on the stability of the peptide salmon calcitonin in aqueous solution
International Journal of Pharmaceutics
Soft drugs based on hydrocortisone: The inactive metabolite approach and its application to steroidal antiinflammatory agents
Pharmaceutical Research
Methods to enhance the complexation efficiency of cyclodextrins
S.T.P. Pharma Sciences
Synthesis of cyclic glycerol ether cyclodextrin derivatives and investigation of their binding properties with drugs
Journal of Inclusion Phenomena
Pharmaceutical applications of β-Cyclodextrin
Pharmaceutical Technology Europe
1998
Cyclodextrins as co-enhancers in dermal and transdermal drug delivery
Pharmazie
Fatty acid extract from cod-liver oil: Activity against herpes simplex virus and enhancement of transdermal delivery of acyclovir in-vitro
Pharmacy and Pharmacology Communications
The effect of water-soluble polymers on the aqueous solubility and complexing abilities of β-cyclodextrin
International Journal of Pharmaceutics
Effect of cod-liver oil extract on the buccal permeation of ergotamine tartrate
Proceedings of the Controlled Release Society
Increasing the cyclodextrin complexation of drugs and drug biovailability through addition of water-soluble polymers
Pharmazie
Cyclodextrins: New drug delivery systems in dermatology
International Journal of Dermatology
Aqueous hydrocortisone mouthwash solution: Clinical evaluation
Acta Odontologica Scandinavica
Cyclodextrin solubilization of ETH-615, a zwitterionic drug
Drug Development and Industrial Pharmacy
Stabilisation of ionic drugs through complexation with non-ionic and ionic cyclodextrins
International Journal of Pharmaceutics
Co-administration of a water-soluble polymer increases the usefulness of cyclodextrins in solid oral dosage forms
Pharmaceutical Research
Effect of the cod-liver oil extract on the buccal permeation of ionized and nonionized forms of ergotamine using the keratinized epithelial-free membrane of hamster cheek pouch mucosa
International Journal of Pharmaceutics
1997
Effect of cyclodextrins on topical drug delivery to the eye
Drug Development and Industrial Pharmacy
Unsaturated glycerol monoethers as novel skin penetration enhancers
Pharmazie
Effect of various marine lipids on transdermal drug delivery - in vitro evaluation
Bollettino Chimico Farmaceutico
Cyclodextrin solubilization of water-soluble drugs: Calcipotriol and EB-1089
Pharmazie
Formulation and testing of methazolamide cyclodextrin eye drop solutions
Journal of Controlled Release
1996
Potentiation of anticancer effects of microencapsulated carboplatin by hydroxypropyl α-cyclodextrin
Journal of Controlled Release
Dexamethasone-cyclodextrin-polymer co-complexes in aqueous eye drops: Aqueous humor pharmacokinetics in humans
Investigative Ophthalmology and Visual Science
The effect of water-soluble polymers on aqueous solubility of drugs
International Journal of Pharmaceutics
Design and in vivo testing of 17β-estradiol-HPβCD sublingual tablets
Pharmazie
The influence of water-soluble polymers and pH on hydroxypropyl-β-cyclodextrin complexation of drugs
Drug Development and Industrial Pharmacy
Pharmaceutical applications of cyclodextrins. 1. Drug solubilization and stabilization
Journal of Pharmaceutical Sciences
Effects of cyclodextrins and polymers on transdermal drug delivery
Proceedings of the Controlled Release Society
Effects of cyclodextrins and polymers on topical drug delivery to the eye - Evaluations in humans
Proceedings of the Controlled Release Society
Topically effective acetazolamide eye-drop solution in man
Pharmaceutical Sciences
Formulation and clinical evaluation of a hydrocortisone solution for the treatment of oral disease
International Journal of Pharmaceutics
1995
Formulation development for a zidovudine chemical delivery system 1. Parenteral dosage forms
International Journal of Pharmaceutics
Improved acitretin delivery through hairless mouse skin by cyclodextrin complexation
International Journal of Pharmaceutics
Fatty acids from cod-liver oil as skin penetration enhancers
Pharmazie
Preparation, characterization, and anesthetic properties of 2- hydroxypropyl-β-cyclodextrin complexes of pregnanolone and pregnenolone in rat and mouse
Journal of Pharmaceutical Sciences
The effect of polyvinylpyrrolidone on cyclodextrin complexation of hydrocortisone and its diffusion through hairless mouse skin
International Journal of Pharmaceutics
Formulation development for a zidovudine chemical delivery system 2. Towards oral and non-parenteral dosage forms
International Journal of Pharmaceutics
1994
The influence of 2-hydroxypropyl-β-cyclodextrin on diffusion rates and transdermal delivery of hydrocortisone
Drug Development and Industrial Pharmacy
The pharmacokinetics and transdermal delivery of loteprednol etabonate and related soft steroids
Advanced Drug Delivery Reviews
The effect of hydroxypropyl methylcellulose on the release of dexamethasone from aqueous 2-hydroxypropyl-β-cyclodextrin formulations
International Journal of Pharmaceutics
2-Hydroxypropyl-β-cyclodextrin in topical carbonic anhydrase inhibitor formulations
European Journal of Pharmaceutical Sciences
Topically effective ocular hypotensive acetazolamide and ethoxyzolamide formulations in rabbits
Journal of Pharmacy and Pharmacology
The effect of water-soluble polymers on drug-cyclodextrin complexation
International Journal of Pharmaceutics
Effect of cyclodextrins on the degradation of cortisone acetate, oestradiol benzoate and prednicarbate in aqueous solution
S.T.P. Pharma Sciences
The influence of cyclodextrins on the stability of cephalotin and aztreonam in aqueous solutions
Pharmazie
The effect of polyvinylpyrrolidone and hydroxypropyl methylcellulose on HPβCD complexation of hydrocortisone and its permeability through hairless mouse skin
European Journal of Pharmaceutical Sciences
1993
Cyclodextrin complexation of NSAIDs: Physicochemical characteristics
European Journal of Pharmaceutical Sciences
The effect of cyclodextrins on the solubility and stability of medroxyprogesterone acetate and megestrol acetate in aqueous solution
International Journal of Pharmaceutics
Topical delivery of acetazolamide for psoriasis
Acta Dermato-Venereologica
1992
Stabilizing effect of tris(hydroxymethyl)aminomethane on N-nitrosoureas in aqueous solutions [1]
Journal of Pharmaceutical Sciences
Improved delivery through biological membranes. XLV. Synthesis, physical-chemical evaluation, and brain uptake studies of 2-chloroethyl nitrosourea delivery systems
Pharmaceutical Research
Effect of various cyclodextrins on solution stability and dissolution rate of doxorubicin hydrochloride
International Journal of Pharmaceutics
The stability of aspartame in aqueous solutions
Acta Pharmaceutica Nordica
Metabolism, distribution, and transdermal permeation of a soft corticosteroid, loteprednol etabonate
Pharmaceutical Research
Preparation and physical evaluation of microcapsules of hydrophilic drug-cyclodextrin complexes
Journal of Microencapsulation
Interactions between preservatives and 2-hydroxypropyl-β-cyclodextrin
Drug Development and Industrial Pharmacy
Degradation of tauromustine (TCNU) in aqueous solutions
Acta Pharmaceutica Nordica
Estramustine: Hydrolysis, solubilization, and stabilization in aqueous solutions
International Journal of Pharmaceutics
1991
Stabilization of aspartame by cyclodextrins
International Journal of Pharmaceutics
2-Hydroxypropyl-β-cyclodextrin: Properties and usage in pharmaceutical formulations
PZ Wissenschaft
Cyclodextrin-accelerated degradation of β-lactam antibiotics in aqueous solutions
International Journal of Pharmaceutics
The effects of cyclodextrins on transdermal delivery of drugs
European Journal of Pharmaceutics and Biopharmaceutics
Solubilization and stabilization of a benzylpenicillin chemical delivery system by 2-hydroxypropyl-β-cyclodextrin
Pharmaceutical Research
Solubilization and stabilization of drugs through cyclodextrin complexation
Acta Pharmaceutica Nordica
1990
Comparative study on inclusion complexation of acetylsalicylic acid, cholecalciferol and melphalan with β- and γ-cyclodextrin and some of their derivatives
Acta Pharmaceutica Nordica
The effect of 2-hydroxypropyl-β-cyclodextrin on the simultaneous dissolution and degradation of chlorambucil
International Journal of Pharmaceutics
Degradation of lomustine (CCNU) in aqueous solutions
International Journal of Pharmaceutics
Novel central nervous system targeted semisynthetic penicillins
Drug Design and Delivery
The effect of phosphine oxides on transdermal delivery
Acta Pharmaceutica Nordica
1989
Effect of oleic acid on diffusion of drugs through hairless mouse skin
Acta Pharmaceutica Nordica
Effect of choline esters and oleic acid on the penetration of acyclovir, estradiol, hydrocortisone, nitroglycerin, retinoic acid and trifluorothymidine across hairles mouse skin in vitro
Acta Pharmaceutica Nordica
The effects of 2-hydroxypropyl-β-cyclodextrin on the solubility and stability of chlorambucil and melphalan in aqueous solution
International Journal of Pharmaceutics
Effects of 2-hydroxypropyl-β-cyclodextrin on the aqueous solubility of drugs and transdermal delivery of 17β-estradiol
Acta Pharmaceutica Nordica
1988
Improved delivery through biological membranes XXXI: Solubilization and stabilization of an estradiol chemical delivery system by modified β-cyclodextrins
Journal of Pharmaceutical Sciences
1987
Trifluorothymidine: potential non-invasive diagnosis of herpes simplex infection using 19F nuclear magnetic resonance in a murine hepatitis model
Journal of Virological Methods
The effect of vehicle additives on the transdermal delivery of nitroglycerin
Pharmaceutical Research
1985
The effect of ionization on partition coefficients and topical delivery
Acta Pharmaceutica Suecica
1984
Synthesis and evaluation of novel lidocaine sulfur analogs
International Journal of Pharmaceutics
Soft drugs VI. The application of the inactive metabolite approach for design of soft β-blockers
Pharmaceutical Research
1981
Improved delivery through biological membranes IX: Kinetics and mechanism of hydrolysis of methylsulfinylmethyl 2-acetoxybenzoate and related aspirin prodrugs
Journal of Pharmaceutical Sciences
Improved delivery through biological membranes VIII: Design, synthesis, and in vivo testing of true prodrugs of aspirin
Journal of Pharmaceutical Sciences
Improved delivery through biological membranes X: Percutaneous absorption and metabolism of methylsulfinylmethyl 2-acetoxybenzoate and related aspirin prodrugs
Journal of Pharmaceutical Sciences
Keywords for Specialisation:
Nanomedicine
Cyclodextrin
Solubility
Bioavailability
Mucosa
Ophtalmic drug delivery
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